1)  Diltiazem
地尔硫婙
2)  minoxidil
米诺地尔
1.
Inhibition on the Proliferation of Hypertrophic Scar Fibroblasts by Minoxidil;
米诺地尔对增生性瘢痕成纤维细胞增殖的影响
2.
Determination of content of minoxidil of compound minoxidil solution;
复方米诺地尔溶液中米诺地尔的含量测定
3.
Preparation and Quality Control of Minoxidil Gel;
米诺地尔凝胶的制备及质量控制
3)  trapidil
曲匹地尔
1.
Improved synthesis of trapidil;
曲匹地尔的合成工艺改进
2.
Effect of Trapidil on the Expression of Matrix Metalloproteinase-2 in Rabbits Aorta After Balloon Injury;
曲匹地尔对兔主动脉球囊损伤后血管壁基质金属蛋白酶-2表达的影响
3.
The Effect of Trapidil on Intimal Hyperplasia of Autografted Vein of Rats;
曲匹地尔对大鼠自体移植静脉内膜增生的影响
4)  nicorandil
尼可地尔
1.
Determination of Nicorandil Based on Its Polarographic Catalytic Wave;
尼可地尔的极谱催化波法测定
2.
Determination of Nicorandil Based on Cation Surfactant Enhancement by Single Sweep Oscillopolarography;
表面活性剂增敏单扫描示波极谱法测定尼可地尔
3.
Effects of ischemic postconditioning and preconditioning induced by Nicorandil on myocardial ischemia/reperfusion injury in isolated rat heart;
尼可地尔后处理联合预处理对离体心肌缺血/再灌注的作用研究
5)  Urapidil
乌拉地尔
1.
Determination of Urapidil by Flow Injection Chemiluminescence;
流动注射-化学发光法测定乌拉地尔
2.
Determination of Urapidil by HPLC;
新药乌拉地尔含量的高效液相色谱法测定
3.
Comparison of clinical efficacy between urapidil and other vasodilators in acute left heart failure;
乌拉地尔治疗急性左心衰竭与其它血管扩张剂疗效比较
6)  naftopidil
萘哌地尔
1.
Determination of naftopidil in human serum by HPLC-fluorescence and study on its pharmacokinetics in healthy volunteers;
高效液相色谱-荧光检测法测定萘哌地尔血药浓度及其在健康人体的药代动力学研究
2.
Evaluation of therapeutic effect of naftopidil in patients with mild to moderate hypertension;
评价萘哌地尔治疗轻中度高血压的临床疗效
3.
The efficacy of naftopidil in treatment of female urethral syndrome;
萘哌地尔治疗女性尿道综合征初探
参考词条
补充资料:地尔硫
分子式:C22H26N2O4S·HCl
分子量:450.98
CAS号:33286-22-5

性质:白色结晶或结晶性粉末。熔点187-188℃。易溶于水、甲醇、氯仿,难溶于无水乙醇,不溶于苯。无臭,味苦。

制备方法:由2-氨基硫酚与对甲氧苯基环氧丙酸乙酯缩合得2-(4-甲氧基苯基)-3-羟基-1,5-苯并硫氮杂 -4(5H)-酮。再经酰化、与二甲氨基氯乙烷缩合、成盐制得硫氮卓酮。

用途:钙通道阻滞药,用于室上性心律失常、心绞痛、老年人高血压等。本品为冠脉扩张药,对心绞痛有效。用于运动性绞痛及陈旧性心肌梗塞引起的心绞痛治疗。本品对雌小鼠口服LD50为640毫克/公斤,雄大鼠口服LD50为560毫克/公斤。

说明:补充资料仅用于学习参考,请勿用于其它任何用途。