1) In vivo knockdown
体内活性抑制
3) in vitro inhibition activity
体外抑制活性
1.
The in vitro inhibition activity of the lipid-soluble epigallocatechin-3-O-gallate-4 -palmitate on ovarian cancer cells HO-8910 was investigated and compared with that of green tea polyphenols and lipophilic tea polyphenol.
药理学实验考察并比较了脂溶性的表没食子儿茶素-3-O-没食子酸-4'-棕榈酸酯、水溶性的绿茶多酚和脂溶性茶多酚对人卵巢癌HO-8910细胞株的体外抑制活性。
4) in vivo Inhibition
活体抑制
5) inhibitory activity
抑制活性
1.
Synthesis and HIV-1 reverse transcriptase inhibitory activity of 3,4-substituted quinolinone derivatives
3,4-取代喹啉酮类衍生物的合成及其对HIV-1逆转录酶的抑制活性
2.
Primary results showed that some of the compounds displayed potential inhibitory activity at a concentration ranging from 0.
2 mmol/L时部分化合物对该酶有较好的抑制活性。
3.
Various kinds of N-substituted pseudo-aminosugars derivatives,which show more potent inhibitory activity against α-glycosidase than the parent compounds,have been synthesized by chemical modification of pseudo-aminosugars.
井冈霉醇胺、井冈霉胺和井冈胺等假氨基糖类物质是新型的α 糖苷酶抑制剂,对其进行化学修饰可以得到糖苷酶抑制活性更强的N 取代假氨基糖衍生物。
6) inhibiting activity
抑制活性
1.
Synthesis, quantitative structure-activity relationship (QSAR) study of inhibiting activity against Sphaerotheca fuliginea and molecular design of acetophenone oxime derivatives based on quantitative structure-activity relationship were performed.
介绍苯乙酮肟醚类化合物的合成、瓜类白粉病抑制活性的定量构效关系(QSAR)研究以及基于QSAR研究结果的新化合物设计、合成和生测,尝试了农药先导合理设计流程在具有瓜类白粉病抑制活性的苯乙酮肟醚类化合物设计中的应用。
2.
According to the result of biological experiments,2-(4,6-dimethoxy-pyrimidin-2-yloxy)-N-het/aryl-benzylamine derivatives were found to have the inhibiting activity of acetolactate synthase(ALS),and the relationship between these compounds and their activity was studied by 3D-QSAR:CoMFA and CoM-SIA.
生物活性测试结果表明,2-嘧啶氧基-N-芳基苄胺类化合物对ALS具有一定的抑制活性。
3.
When acted with equal proportion of Papain , the inhibiting activity of CPI lost completely; CD spectrum changed remarkably and the content of α-helix declined.
水稻巯基蛋白酶抑制剂(CPI)圆二色性谱(CD)显示206nm和222nm处的双负峰,CPI分子以α 螺旋构象为主;当CPI与木瓜蛋白酶等摩尔结合后,CPI完全丧失抑制活性,复合物CD谱发生显著变化,α 螺旋含量降低。
补充资料：体内
分子式：
CAS号：
性质：常指实验观察中的事件或酶反应以正常途径发生，即在一个生物活体之内进行。
CAS号：
性质：常指实验观察中的事件或酶反应以正常途径发生，即在一个生物活体之内进行。
说明：补充资料仅用于学习参考，请勿用于其它任何用途。
参考词条