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1)  5-aza-cytidine
组蛋白脱乙酰化酶抑制剂
1.
DNA methyltransferase (DNMT) inhibitor, 5-aza-cytidine (5-aza-C), was widely studied because DNA hypomethylation induced the re-activation of tumor suppressor genes that were silenced by methylation-mediated mechanisms, could inhibit proliferation and induce differentiation of tumor.
组蛋白脱乙酰化酶抑制剂苯丁酸钠(sodium phenylbutyrate,SPB)通过对组蛋白去乙酰化酶(histone seacetylase,HDAC)的抑制而达到对肿瘤细胞的生长抑制、诱导分化及诱导凋亡的作用。
2)  Histone Deacetylase Inhibitor
组蛋白脱乙酰酶抑制剂
3)  histone deacetylase inhibitor
组蛋白脱乙酰基酶抑制剂
4)  histone deacetylase inhibitors
组蛋白去乙酰酶抑制剂
1.
Progress in the research of histone deacetylase inhibitors;
组蛋白去乙酰酶抑制剂的研究进展
5)  histone deacetylase(HDAC) inhibitor
组蛋白乙酰酶抑制剂
6)  histone deacetylase inhibitors
组蛋白去乙酰化酶抑制剂
1.
Mechanism of histone deacetylase inhibitors for treatment of hematological cancer and their clinical research;
组蛋白去乙酰化酶抑制剂治疗血液系统肿瘤的作用机制及临床应用
2.
Molecular mechanism of p21~(WAF1/CIP1) expression induced by histone deacetylase inhibitors in HeLa cell line;
组蛋白去乙酰化酶抑制剂诱导H eLa细胞p21~(WAF1/CIP1)表达的分子机制研究
3.
Mechanism of regulating multidrug resistances by histone deacetylase inhibitors in tumor cells;
组蛋白去乙酰化酶抑制剂调节肿瘤细胞多药耐药性的机制
补充资料:多巴脱羧酶抑制剂
分子式:
CAS号:

性质:能够抑制多巴脱羧酶活性的一类化学物质,如在曲霉和链霉菌发酵液中发现的一类异黄酮,能够非特异性地抑制多巴脱羧酶活性,对自发性高血压的大鼠有降压作用,活性大小与α-甲基多巴胺相当。

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