1) inhibitory effects on NO production
抑制NO释放活性
2) inhibitory effect of NO production
抑制巨嗜细胞嗜放NO活性
3) inhibitory activity
抑制活性
1.
Synthesis and HIV-1 reverse transcriptase inhibitory activity of 3,4-substituted quinolinone derivatives
3,4-取代喹啉酮类衍生物的合成及其对HIV-1逆转录酶的抑制活性
2.
Primary results showed that some of the compounds displayed potential inhibitory activity at a concentration ranging from 0.
2 mmol/L时部分化合物对该酶有较好的抑制活性。
3.
Various kinds of N-substituted pseudo-aminosugars derivatives,which show more potent inhibitory activity against α-glycosidase than the parent compounds,have been synthesized by chemical modification of pseudo-aminosugars.
井冈霉醇胺、井冈霉胺和井冈胺等假氨基糖类物质是新型的α 糖苷酶抑制剂,对其进行化学修饰可以得到糖苷酶抑制活性更强的N 取代假氨基糖衍生物。
4) inhibiting activity
抑制活性
1.
Synthesis, quantitative structure-activity relationship (QSAR) study of inhibiting activity against Sphaerotheca fuliginea and molecular design of acetophenone oxime derivatives based on quantitative structure-activity relationship were performed.
介绍苯乙酮肟醚类化合物的合成、瓜类白粉病抑制活性的定量构效关系(QSAR)研究以及基于QSAR研究结果的新化合物设计、合成和生测,尝试了农药先导合理设计流程在具有瓜类白粉病抑制活性的苯乙酮肟醚类化合物设计中的应用。
2.
According to the result of biological experiments,2-(4,6-dimethoxy-pyrimidin-2-yloxy)-N-het/aryl-benzylamine derivatives were found to have the inhibiting activity of acetolactate synthase(ALS),and the relationship between these compounds and their activity was studied by 3D-QSAR:CoMFA and CoM-SIA.
生物活性测试结果表明,2-嘧啶氧基-N-芳基苄胺类化合物对ALS具有一定的抑制活性。
3.
When acted with equal proportion of Papain , the inhibiting activity of CPI lost completely; CD spectrum changed remarkably and the content of α-helix declined.
水稻巯基蛋白酶抑制剂(CPI)圆二色性谱(CD)显示206nm和222nm处的双负峰,CPI分子以α 螺旋构象为主;当CPI与木瓜蛋白酶等摩尔结合后,CPI完全丧失抑制活性,复合物CD谱发生显著变化,α 螺旋含量降低。
5) inhibition of telomerase activity
活性抑制
1.
BACKGROOND&AIM: To study the inhibition of telomerase activity in melanoma A 375 cells by arsenic trioxide(As 2 O 3 ).
结果 :As2O3 对人恶性黑色素瘤A375 细胞端粒酶活性抑制有明显的浓度和时间依赖关系。
6) inhibitory activities
抑制性活
补充资料：促黑激素释放抑制因子
分子式：
CAS号：
性质：又称促黑激素释放抑制因子。自下丘脑分离或入工合成制得，已发现的两种化学结构分别是Pro-Leu-Gly-NH2三肽和Pro-His-Phe-Arg-Gly-NH2五肽。MRIF是下丘脑所分泌的激素释放抑制因子之一，其生理功能是抑制垂体促黑色细胞激素(MSH)的释放，用于治疗抑郁和帕金森氏病。
CAS号：
性质：又称促黑激素释放抑制因子。自下丘脑分离或入工合成制得，已发现的两种化学结构分别是Pro-Leu-Gly-NH2三肽和Pro-His-Phe-Arg-Gly-NH2五肽。MRIF是下丘脑所分泌的激素释放抑制因子之一，其生理功能是抑制垂体促黑色细胞激素(MSH)的释放，用于治疗抑郁和帕金森氏病。
说明：补充资料仅用于学习参考，请勿用于其它任何用途。
参考词条