1) Raf inhibitor
Raf阻断剂
1.
Raf inhibitors have been developed and some are being evaluated in clinical trials.
一些Raf阻断剂正在临床试验中,因特定Raf基因过表达而发生的恶性肿瘤很可能会对raf蛋白的阻断剂敏感。
2) Blocking agent
阻断剂
1.
Lycopene can be biosynthesized by adding blocking agents to Blakeslea trispora which can produce β-carotenewith high yield or by employing mutant strain of Blakeslea trispora.
利用β-胡萝卜素高产菌株三孢布拉氏霉菌(Blakeslea trispora)发酵生产番茄红素过程中,可通过突变菌株或中途加入阻断剂的方法,将代谢控制在番茄红素水平。
2.
Methods 5 HT 1 receptor stimulant 1 (3 chorophenyl) piperazine,5 HT 2 receptor stimulant α CH 3 5 HT,5 HT 2 receptor blocking agent-Methiothepin mesylate and 5 HT 2 receptor stimulant-Retanserine were respectively injected into the lateral ventricle of rat with morphine dependence,and then the effect on morphine withdrawal syndromes was observed.
方法 分别给吗啡依赖大鼠侧脑室注射 5 HT1受体激动剂 1 (3 chlorophenyl)piperazine(简称m cpp)、5 HT2 受体激动剂α CH3 5 HT和 5 HT1受体阻断剂Methiothepinmesylate、5 HT2 受体阻断剂Retanserine ,观察对吗啡戒断反应的影响。
3) β-blocker
β-阻断剂
1.
Chemical Ionization (CI) Application to the Confirmation of β-blockers;
化学电离(CI)在β-阻断剂确证中的应用研究
2.
Studies on the Analysis of β-blockers and Their Metabolites in Urine by Gas Chromatography (Ⅲ)──Analysis of Five β-Blockers and Their Metabolites in Rats' Urine by Solid-phase Extraction and GC/MS;
β-阻断剂及其代谢产物的气相色谱分析研究(Ⅲ)──用固相提取及GC/MS法分析大鼠尿中5种β-阻断剂及其代谢物
4) inhibitor
[英][in'hibitə] [美][ɪn'hɪbətɚ]
阻断剂
1.
Effects of p38 inhibitor on expression of IL-6 stimulated by mechanical pressure in HPLF;
p38丝裂原激活蛋白阻断剂对机械压力诱导人牙周膜成纤维细胞表达白介素-6的影响
2.
Objective To observe the effect of intra-articular injection of SB203580,a selective p38 mitogen-activated protein kinase inhibitor,on the expression of matrix metalloproteinase(MMP)-3,MMP-13 in a rat model of osteoarthritis(OA) and to explore the relationship between the MMP-3/MMP-13 expressions and the severity of OA.
目的观察p38信号转导途径阻断剂SB203580经关节腔注射对实验性鼠膝骨关节炎基质金属蛋白酶(MMP)-3、MMP-13表达的影响,探讨MMP-3、MMP-13表达与创伤性软骨退变之间的关系。
3.
Methods Thirteen kind inhibitors which possibly block the cytotoxic effects of palmitic acid on human umbilical vein endothelial cell (HUVEC)were selected.
结果 ①一氧化氮合酶阻断剂 (-N 硝基L 精氨酸 ,L NNA)能部分阻断PA引起血管内皮细胞死亡 [1 5 μmol LL NNA+2 0 0 μmol LPA组与 2 0 0 μm LPA单独作用组比较细胞生存率增加了 4 3。
6) blocker
[英]['blɔkə] [美]['blɑkɚ]
阻断剂
1.
Research progress in N-type calcium channel and its blockers;
N-型钙通道及其阻断剂研究进展
2.
Theω-conotoxin MⅦA from Conus magus is a specific and selective blocker of N-type voltage-sensi-tive calcium channels.
其中,ω-芋螺毒素MⅦA来自致幻芋螺(Conusmagus),是一种高选择性的N-型电压敏感型Ca2+通道阻断剂。
补充资料:5-羟色胺受体阻断剂
分子式:
CAS号:
性质:5-羟色胺(5-HT)是重要的神经递质,也是一种自身活性物质。5-HT通过与靶细胞膜上的5-HT受体结合并诱发生物效应。5-HT受体可分为5-HT1A,5-HT1B,5-HT1C,5-HT2,5-HT3。5-HT受体阻断药大致有以下几类,(1)麦角酸的衍生物如麦解酰二乙胺等;(2)组胺H1受体阻断药如赛庚啶等;(3)吩噻嗪类如氯丙嗪等;(4)肾上腺素α-受体阻断药如酚苄明等。常用于实验室研究、较为特异的5-HT受体阻断剂有麦角苄脂、米安色林、苯噻啶等。
CAS号:
性质:5-羟色胺(5-HT)是重要的神经递质,也是一种自身活性物质。5-HT通过与靶细胞膜上的5-HT受体结合并诱发生物效应。5-HT受体可分为5-HT1A,5-HT1B,5-HT1C,5-HT2,5-HT3。5-HT受体阻断药大致有以下几类,(1)麦角酸的衍生物如麦解酰二乙胺等;(2)组胺H1受体阻断药如赛庚啶等;(3)吩噻嗪类如氯丙嗪等;(4)肾上腺素α-受体阻断药如酚苄明等。常用于实验室研究、较为特异的5-HT受体阻断剂有麦角苄脂、米安色林、苯噻啶等。
说明:补充资料仅用于学习参考,请勿用于其它任何用途。
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