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1)  validoxylamine A
井冈羟胺A
1.
Preparation and characterization of the trehalase inhibitor validoxylamine A;
海藻糖酶抑制剂井冈羟胺A的制备与表征
2.
Forty new compounds of validoxylamine A derivatives were prepared based on validoxylamine A as the leading compound.
井冈霉素是高效、安全和作用机制独特的无公害生物农药,其水解产物井冈羟胺A是已知天然海藻糖酶抑制剂中抑酶活性最高的化合物之一。
3.
This research focused on the chemical modification of natural compound validoxylamine A and small-molecular compound hexahydropyridazine.
本论文分别对天然化合物井冈羟胺A和小分子化合物六氢哒嗪进行结构修饰,合成了一系列新化合物,并对其中部分进行了生物活性测试。
2)  jinggangamines
井冈羟胺
3)  7-O-chrysanthemyl validoxylamine A
7-O-菊酰基井冈羟胺A
1.
Synthesis of 7 -O-chrysanthemyl validoxylamine A;
7 -O-菊酰基井冈羟胺A的合成
4)  valienamine
井冈胺
1.
It has a low price while valienamine, an important intermediate of medicine, is much more expensive.
井冈胺是井冈霉素的组成部分,是重要的医药中间体,其销售价格是井冈霉素的几十倍。
2.
Validamycins have been one of the most popular and economical biopesticides in China, by microbial transformation of which validoxylamine A and valienamine can be produced.
井冈霉素目前已成为我国最经济最受欢迎的生物农药之一,用微生物转化法分解井冈霉素可以得到井冈霉亚基胺A和井冈胺,前者对海藻糖酶有强烈的抑制作用,有望开发成为新型生物杀虫剂,而后者是一种糖苷酶抑制剂,也可作为合成降糖药的原料。
3.
In this paper, the inhibition of valienamine and validamine on porcine intestinal suc.
本实验室以井冈霉素为原料,采用微生物催化技术,得到了环醇类物质井冈胺、井冈霉胺和井冈霉亚基胺A。
5)  validamine
井冈霉胺
1.
In our lab, validamycins were used as raw material, cyclitol compounds such as vaienamine, validamine, and validoxylamine A were obtained by microbial catalysis.
本实验室以井冈霉素为原料,采用微生物催化技术,得到了环醇类物质井冈胺、井冈霉胺和井冈霉亚基胺A。
6)  valiolamine
井冈霉醇胺
1.
N-Substituted chemical modification of valiolamine,as well as the inhibitory activity of these compounds against porcine and rat intestinal maltase and surase are discussed in detail.
井冈霉醇胺、井冈霉胺和井冈胺等假氨基糖类物质是新型的α 糖苷酶抑制剂,对其进行化学修饰可以得到糖苷酶抑制活性更强的N 取代假氨基糖衍生物。
补充资料:阴冈
1.山冈的北边。
说明:补充资料仅用于学习参考,请勿用于其它任何用途。
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